Palladium-catalyzed intramolecular C-H activation/C-C bond formation: A straightforward synthesis of phenanthridines
Document Type
Article
Publication Date
11-18-2011
Abstract
The palladium-catalyzed intramolecular C-H activation/C-C cross-coupling has been developed for a straightforward and efficient synthesis of phenanthridines. With Pd(OAc) 2 (4 mol %) as the catalyst, PCy 3 (8 mol %) as the ligand, and Cs 2CO 3 as the base, this protocol was applied to synthesize a small library of phenanthridine derivatives in good yields in THF. © 2011 American Chemical Society.
Publication Source (Journal or Book title)
Journal of Organic Chemistry
First Page
9507
Last Page
9513
Recommended Citation
Peng, J., Chen, T., Chen, C., & Li, B. (2011). Palladium-catalyzed intramolecular C-H activation/C-C bond formation: A straightforward synthesis of phenanthridines. Journal of Organic Chemistry, 76 (22), 9507-9513. https://doi.org/10.1021/jo2017108
COinS